SCHEMBL8105023

SCHEMBL8105023

N#Cc1ccc(Cc2cnc(Cc3ccc(-c4ccccc4)cc3CN)[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 11/20 0.52
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
AOC3 Q16853 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
EP300 Q09472 1/20 0.36
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8305243 0.99 BRS3 (0.51) BRS3CYP11B1CYP11B2HRH3NOS3
SCHEMBL8097357 0.89 BRS3 (0.51) BRS3CYP11B1CYP11B2HRH3GABRA1
Hydrochloric Acid SCHEMBL8307882 0.88 BRS3 (0.50) BRS3CYP11B1CYP11B2HRH3GABRA1
SCHEMBL8106552 0.87 BRS3 (0.49) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7927535 0.86 BRS3 (0.52) BRS3CYP11B1CYP11B2HRH3GABRA1
Hydrochloric Acid SCHEMBL8306714 0.86 BRS3 (0.48) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7919393 0.85 BRS3 (0.62) BRS3CYP11B1CYP11B2HRH3AOC3
Hydrochloric Acid SCHEMBL8521500 0.84 BRS3 (0.61) BRS3CYP11B1CYP11B2HRH3AOC3
SCHEMBL8305740 0.82 BRS3 (0.59) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7924356 0.81 BRS3 (0.72) BRS3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP claimed
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP claimed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO claimed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO claimed
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP disclosed
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO disclosed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed