SCHEMBL8106552

SCHEMBL8106552

CCCCc1cc(-c2ccccc2)ccc1Cc1ncc(Cc2ccc(C#N)cc2)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 12/20 0.49
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
HRH3 Q9Y5N1 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8306714 0.99 BRS3 (0.48) BRS3TSHRHSD17B10CYP11B1CYP11B2
SCHEMBL8097357 0.94 BRS3 (0.51) BRS3TSHRHSD17B10CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL8307882 0.93 BRS3 (0.50) BRS3TSHRHSD17B10CYP11B1CYP11B2
SCHEMBL8105023 0.87 BRS3 (0.52) BRS3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8305243 0.86 BRS3 (0.51) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7927535 0.84 BRS3 (0.52) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7919393 0.83 BRS3 (0.62) BRS3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8521500 0.82 BRS3 (0.61) BRS3CYP11B1CYP11B2HRH3
SCHEMBL8107069 0.79 BRS3 (0.51) BRS3TSHRHSD17B10CYP11B1CYP11B2
SCHEMBL7924356 0.79 BRS3 (0.72) BRS3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP claimed
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP claimed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO claimed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO claimed
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP disclosed
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO disclosed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed