SCHEMBL8106035

SCHEMBL8106035

CC(C)CC(=O)Nc1ccc(-c2nc(N)cc(CS(C)(=O)=O)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.52
PIK3CA P42336 5/20 0.47
PIK3CD O00329 4/20 0.47
MTOR P42345 3/20 0.46
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
NPC1 O15118 3/20 0.45
ALDH1A1 P00352 2/20 0.45
GFER P55789 1/20 0.45
ADORA2A P29274 2/20 0.44
ADORA3 P0DMS8 1/20 0.44
ADORA1 P30542 1/20 0.44
HPGD P15428 3/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 2/20 0.43
SENP7 Q9BQF6 1/20 0.43
CASP3 P42574 1/20 0.43
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101524 0.87 MEN1 (0.54) PIK3CAPIK3CDMTORRAB9ASMN1; SMN2
SCHEMBL8093349 0.87 PIK3CD (0.48) PIK3CAPIK3CDMTORSMN1; SMN2ALDH1A1
SCHEMBL8106030 0.86 PIK3CA (0.47) PIK3CAPIK3CDMTORRAB9ASMN1; SMN2
SCHEMBL8101525 0.85 TP53 (0.51) PIK3CAPIK3CDMTORRAB9ASMN1; SMN2
SCHEMBL11925797 0.85 PIK3CA (0.49) PIK3CAPIK3CDMTORALDH1A1HPGD
SCHEMBL8213955 0.85 PIK3CA (0.53) PIK3CAPIK3CDMTORLMNA
SCHEMBL8215098 0.84 PIK3CA (0.50) PIK3CAPIK3CDMTORALDH1A1HPGD
SCHEMBL8104034 0.84 MAPT (0.49) PIK3CAPIK3CDMTORALDH1A1HPGD
SCHEMBL8103957 0.84 PIK3CD (0.47) PIK3CAPIK3CDMTORRAB9ASMN1; SMN2
SCHEMBL8109642 0.84 PIK3CA (0.49) PIK3CAPIK3CDMTORALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007749-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed