SCHEMBL8104034

SCHEMBL8104034

CN(C)CC(=O)Nc1ccc(-c2nc(N)cc(CS(C)(=O)=O)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
PIK3CA P42336 6/20 0.47
PIK3CD O00329 6/20 0.47
MTOR P42345 4/20 0.46
TAAR1 Q96RJ0 1/20 0.43
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 2/20 0.40
HPGD P15428 2/20 0.40
KMT2A Q03164 2/20 0.40
MAP4K4 O95819 1/20 0.40
KDR P35968 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101524 0.87 MEN1 (0.54) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8093349 0.87 PIK3CD (0.48) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8101525 0.85 TP53 (0.51) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL11925797 0.85 PIK3CA (0.49) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8214091 0.85 PIK3CA (0.48) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8106035 0.84 PTPN1 (0.52) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8103957 0.84 PIK3CD (0.47) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8086546 0.83 PIK3CD (0.50) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8106107 0.83 CA12 (0.49) MAPTPIK3CAPIK3CDMTORALDH1A1
SCHEMBL8103980 0.83 PIK3CA (0.47) MAPTPIK3CAPIK3CDMTORALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007749-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed