SCHEMBL8106049

SCHEMBL8106049

N#Cc1ccc(Cc2ncc(CNc3cccc(CCc4ccccc4)n3)[nH]2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 4/20 0.46
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
NTRK1 P04629 2/20 0.38
KCNH2 Q12809 1/20 0.37
OPRM1 P35372 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
JAK2 O60674 1/20 0.36
ABL1 P00519 1/20 0.36
INSR P06213 1/20 0.36
LCK P06239 1/20 0.36
CSF1R P07333 1/20 0.36
LYN P07948 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116598 0.84 BRS3 (0.41) BRS3CYP1A2CYP2D6CYP2C19LMNA
SCHEMBL8298317 0.77 BRS3 (0.48) BRS3OPRM1ABCG2CYP19A1
Hydrochloric Acid SCHEMBL8304229 0.76 BRS3 (0.47) BRS3OPRM1ABCG2CYP19A1
SCHEMBL8115034 0.75 GRIN1 (0.38) BRS3CYP1A2CYP2C19LMNAOPRM1
SCHEMBL8120803 0.73 FNTA (0.52) KCNH2
SCHEMBL7461594 0.73 BRS3 (0.48) BRS3EP300
SCHEMBL7919393 0.72 BRS3 (0.62) BRS3CYP19A1GRIN1GRIN2BEP300
Hydrochloric Acid SCHEMBL8004159 0.72 BRS3 (0.48) BRS3EP300
Hydrochloric Acid SCHEMBL8521500 0.71 BRS3 (0.61) BRS3CYP19A1GRIN1GRIN2BEP300
SCHEMBL7924356 0.70 BRS3 (0.72) BRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019391-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO. INC. (US) 2000-07-19 EP disclosed
WO-1999018096-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1999-04-15 WO disclosed