Bromide

Bromide

SCHEMBL8106532

Br.CN1C2C=C(c3cncc4ccc(C5CCCCC5)cc34)CC1CC2

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 5/20 0.42
SLC6A4 known ✓ P31645 5/20 0.42
SLC6A3 known ✓ Q01959 5/20 0.42
HTR6 P50406 1/20 0.36
HRH3 Q9Y5N1 1/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
BACE1 P56817 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
MEN1 O00255 1/20 0.30
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
EGLN1 Q9GZT9 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8106535 1.00 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3HTR6HRH3
SCHEMBL8107623 0.79 SLC6A2 (0.57) SLC6A2SLC6A4SLC6A3HTR6IRAK4
SCHEMBL8107625 0.79 SLC6A2 (0.57) SLC6A2SLC6A4SLC6A3HTR6IRAK4
Bromide SCHEMBL8108934 0.73 HRH3 (0.37) HRH3BACE1IRAK4EGLN1
SCHEMBL5829723 0.67 SLC6A2 (0.53) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL5829382 0.66 SLC6A2 (0.52) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL5829679 0.66 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HTR6
SCHEMBL5829744 0.66 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HTR6
SCHEMBL5829678 0.66 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HTR6
SCHEMBL5829742 0.66 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107307-A PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY (US) 2000-08-22 US disclosed
EP-0969005-A1 Azabicyclic inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 2000-01-05 EP disclosed
WO-1999065492-A1 INHIBITION OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1999-12-23 WO disclosed