SCHEMBL8106554

SCHEMBL8106554

CC(O)C[C@@H]1C[C@@H](O[Si](C)(C)C(C)(C)C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.35
NR1H2 P55055 1/20 0.34
IDO1 P14902 1/20 0.32
PRMT5 O14744 2/20 0.32
WDR77 Q9BQA1 2/20 0.32
CCR2 P41597 2/20 0.31
HTRA1 Q92743 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
VHL P40337 1/20 0.31
ELOC Q15369 1/20 0.31
ELOB Q15370 1/20 0.31
SRC P12931 4/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9595418 1.00 ABCB1 (0.35) ABCB1NR1H2IDO1PRMT5WDR77
SCHEMBL8108567 0.91 ABCB1 (0.34) ABCB1NR1H2CCR2HTRA1
SCHEMBL9595613 0.91 ABCB1 (0.34) ABCB1NR1H2CCR2HTRA1
SCHEMBL8107520 0.90 NR1H2 (0.34) ABCB1NR1H2CCR2SRC
SCHEMBL4669448 0.88 NR1H2 (0.35) ABCB1NR1H2ALDH1A1CHRM2CHRM1
SCHEMBL7451687 0.88 NR1H2 (0.35) ABCB1NR1H2ALDH1A1CHRM2CHRM1
SCHEMBL4669615 0.88 NR1H2 (0.35) ABCB1NR1H2ALDH1A1CHRM2CHRM1
SCHEMBL9596179 0.88 ABCB1 (0.36) ABCB1NR1H2IDO1
SCHEMBL9596361 0.88 ABCB1 (0.36) ABCB1NR1H2IDO1
SCHEMBL12431668 0.87 NR1H2 (0.37) ABCB1NR1H2ALDH1A1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545290-B1 Aminoalkylpyrrolidinylthiocarbapenem derivatives BANYU PHARMA CO LTD (JP) 2000-08-23 EP disclosed
US-5550121-A ANTIBIOTICS BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
EP-0545290-A1 Aminoalkylpyrrolidinylthiocarbapenem derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-09 EP disclosed