SCHEMBL8106701

SCHEMBL8106701

C[C@@H]1CN(c2cccc(OC(F)(F)F)c2)CCN1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.55
CASR P41180 6/20 0.46
KHK P50053 2/20 0.46
ACACB O00763 1/20 0.44
ADRB1 P08588 1/20 0.44
XIAP P98170 1/20 0.44
BIRC2 Q13490 1/20 0.44
PIM1 P11309 1/20 0.44
DHFR P00374 1/20 0.44
FFAR4 Q5NUL3 1/20 0.43
MAPT P10636 2/20 0.42
CHRM2 P08172 2/20 0.41
CHRM1 P11229 1/20 0.41
MLYCD O95822 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5272828 0.91 NOTUM (0.45) NOTUMCASRKHKACACBADRB1
SCHEMBL8108584 0.88 NOTUM (0.44) NOTUMCASRKHKACACBADRB1
SCHEMBL1471079 0.85 MCHR1 (0.44) CASRKHKADRB1XIAPBIRC2
SCHEMBL1005159 0.85 MCHR1 (0.44) CASRKHKADRB1XIAPBIRC2
SCHEMBL1471081 0.85 MCHR1 (0.44) CASRKHKADRB1XIAPBIRC2
SCHEMBL1472870 0.85 NOTUM (0.52) NOTUMCASRACACBPIM1DHFR
SCHEMBL1472865 0.85 NOTUM (0.52) NOTUMCASRACACBPIM1DHFR
Hydrochloric Acid SCHEMBL2244493 0.83 MCHR1 (0.43) CASRKHKADRB1XIAPBIRC2
SCHEMBL2873025 0.83 ADRB1 (0.65) KHKADRB1MAPT
SCHEMBL2873027 0.83 ADRB1 (0.65) KHKADRB1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed