SCHEMBL8109340

SCHEMBL8109340

O=C(O)c1ccc(-c2cnc3ccccc3c2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.68
PDGFRB P09619 3/20 0.59
PDGFRA P16234 3/20 0.59
MAP4K4 O95819 5/20 0.58
CSNK1G2 P78368 1/20 0.58
CLK4 Q9HAZ1 1/20 0.58
MKNK2 Q9HBH9 1/20 0.58
MAP4K5 Q9Y4K4 1/20 0.58
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA9 Q16790 1/20 0.57
FASN P49327 1/20 0.55
PTGES O14684 1/20 0.55
ALOX5 P09917 1/20 0.55
PIK3CD O00329 1/20 0.53
PIK3CA P42336 1/20 0.53
MMP1 P03956 1/20 0.52
MMP9 P14780 1/20 0.52
CYP2A6 P11509 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26613435 0.86 CA12 (0.60) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL12797767 0.84 NPC1 (0.64) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL24621829 0.84 PDGFRB (0.72) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL29375510 0.84 PDGFRB (0.72) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL26829682 0.84 PDGFRB (0.72) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL4130703 0.84 PDGFRB (0.56) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL4123055 0.84 MGAM (0.58) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL12580411 0.83 PDGFRB (0.66) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL12580402 0.83 PDGFRB (0.66) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2
SCHEMBL12580362 0.83 PDGFRB (0.66) MGAMPDGFRBPDGFRAMAP4K4CSNK1G2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1260781-A Indole derivatives having combined 5HT1A, 5HT1B and 5HT1D receptor antagonist activity SMITHKLINE BEECHAM PLC (GB) 2000-07-19 CN disclosed
EP-0975593-A1 INDOLE DERIVATIVES HAVING COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2000-02-02 EP disclosed
WO-1998050358-A1 INDOLE DERIVATIVES HAVING COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed