SCHEMBL8109410

SCHEMBL8109410

O=C(Cl)c1cc(F)cc(C(F)(F)F)c1.O=C(Cl)c1ccc(F)cc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.43
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
VNN1 O95497 3/20 0.39
P2RX1 P51575 1/20 0.37
TMPRSS4 Q9NRS4 1/20 0.37
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
DDR1 Q08345 1/20 0.35
GPBAR1 Q8TDU6 2/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
CSF1R P07333 1/20 0.34
CETP P11597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679186 0.85 CES2 (0.47) CES2KMT2AATMP2RX1TMPRSS4
SCHEMBL7728942 0.84 CETP (0.40) CES2KMT2AATMVNN1CETP
SCHEMBL679313 0.83 CES2 (0.52) CES2VNN1DDR1GPBAR1RXRA
SCHEMBL29593993 0.83 CES2 (0.52) CES2VNN1DDR1GPBAR1RXRA
SCHEMBL8703955 0.79 CES2 (0.41) CES2VNN1TMPRSS4DDR1RXRA
SCHEMBL30518051 0.75 CES2 (0.72) CES2KMT2ATMPRSS4FLT1FLT4
SCHEMBL9230110 0.75 CES2 (0.47) CES2KMT2AATMFLT1FLT4
SCHEMBL937022 0.75 CES2 (0.72) CES2KMT2ATMPRSS4FLT1FLT4
SCHEMBL8701942 0.73 KCNQ3 (0.40) KMT2AATMVNN1
SCHEMBL322157 0.73 CES2 (0.67) CES2P2RX1RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed