SCHEMBL8109957

SCHEMBL8109957

CCN(C=O)OC[C@H]1O[C@@H](n2cnc3c(N)nc(OCCc4ccccc4)nc32)C(O)C1O

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.71
ADORA2B P29275 12/20 0.71
ADORA1 P30542 7/20 0.71
ADORA3 P0DMS8 6/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8102783 0.93 ADORA2A (0.71) ADORA2AADORA2BADORA1ADORA3
SCHEMBL2291656 0.83 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL30862346 0.83 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8115549 0.83 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8109955 0.81 ADORA2A (0.64) ADORA2AADORA2BADORA1ADORA3
SCHEMBL5490949 0.80 ADORA2A (0.73) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8110844 0.79 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8110831 0.79 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL31060329 0.79 ADORA2A (1.00) ADORA2AADORA2BADORA1ADORA3
SCHEMBL2121393 0.79 AHCY (0.66) ADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0515514-B1 2-ARALKOXY AND 2-ALKOXY ADENOSINE DERIVATIVES AS CORONARY VASODILATORS AND ANTIHYPERTENSIVE AGENTS DISCOVERY THERAPEUTICS INC (US) 2000-08-30 EP disclosed
US-RE36494-E 2-aralkoxy and 2-alkoxy adenosine derivatives as coronary vasodilators and antihypertensive agents DISCOVERY THERAPEUTICS, INC. (US) 2000-01-11 US disclosed
US-5140015-A Racemic mixture for inducing an adenosine response in humans and animals WHITBY RESEARCH, INC. (US) 1992-08-18 US disclosed