SCHEMBL8111483

SCHEMBL8111483

Nc1ccc(NCCc2c[nH]c3ccccc23)c(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 12/20 0.58
HTR2A P28223 4/20 0.51
HTR7 P34969 3/20 0.51
HTR6 P50406 3/20 0.51
MPO P05164 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2A6 P11509 1/20 0.51
NFKB1 P19838 1/20 0.51
HTR1D P28221 1/20 0.51
HTR1B P28222 1/20 0.51
HTR2C P28335 1/20 0.51
CTSK P43235 1/20 0.51
CYP2A13 Q16696 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
HTR1A P08908 3/20 0.51
HTT P42858 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17464549 0.87 CDK2 (0.55) CDK2HTR2AHTR7HTR6MPO
SCHEMBL8050581 0.82 CDK2 (0.55) CDK2HTR2AHTR7HTR6HTR1A
SCHEMBL8265688 0.80 MEN1 (0.55) CDK2HTR2AHTR7HTR6HTR1A
SCHEMBL8048284 0.79 HTR2A (0.56) CDK2HTR2AHTR7HTR6MPO
SCHEMBL8263255 0.79 HTR2A (0.65) HTR2AHTR7HTR6MPOCYP1A2
SCHEMBL28384834 0.78 HTR2A (0.66) CDK2HTR2AHTR7HTR6MPO
SCHEMBL4786975 0.78 HTR2A (0.55) CDK2HTR2AHTR7HTR6MPO
SCHEMBL18783077 0.77 CDK2 (0.55) CDK2HTR2ACYP1A2HTR1AHTT
SCHEMBL8041168 0.76 HTR2A (0.56) CDK2HTR2AHTR7HTR6CYP1A2
SCHEMBL8041585 0.74 POLB (0.59) CDK2HTR2AHTR7HTR6MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008132155-A2 INHIBITORS OF THE BINDING BETWEEN HDM2 AND THE PROTEASOME JANSSEN PHARMACEUTICA NV (BE) 2008-11-06 WO disclosed