SCHEMBL8112784

SCHEMBL8112784

N=C(N)NCCC[C@H](C(=O)NCC(=O)O)N(Cc1ccccc1)C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.41
CNR2 P34972 4/20 0.37
EPOR P19235 2/20 0.36
MME P08473 3/20 0.36
ALDH1A1 P00352 1/20 0.36
ACE P12821 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8120085 0.94 CNR1 (0.36) CNR1CNR2EPOR
SCHEMBL8122513 0.94 HDAC3 (0.37) CNR1CNR2EPORMME
SCHEMBL8127029 0.94 NPY1R (0.41) CNR1CNR2EPOR
SCHEMBL8122704 0.93 TPSAB1 (0.36) CNR1CNR2EPOR
SCHEMBL8126149 0.93 TDP1 (0.45) CNR1EPOR
SCHEMBL8112714 0.93 MEN1 (0.42) CNR1CNR2
SCHEMBL8113179 0.92 CNR1 (0.41) CNR1CNR2EPOR
SCHEMBL8113195 0.92 CNR1 (0.34) CNR1CNR2EPORMME
SCHEMBL8529383 0.91 EPOR (0.38) CNR1EPORMME
SCHEMBL8128254 0.90 TPSAB1 (0.38) CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed
EP-0680469-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1995-11-08 EP disclosed
WO-1994017035-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME DR. KARL THOMAE GMBH (DE) 1994-08-04 WO disclosed