SCHEMBL8112944

SCHEMBL8112944

COc1ccccc1-n1nnnc1Br

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 7/20 0.60
ALDH1A1 P00352 8/20 0.58
TSHR P16473 2/20 0.48
HTT P42858 2/20 0.48
HPGD P15428 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ALOX15 P16050 1/20 0.43
P2RX7 Q99572 1/20 0.41
MGLL Q99685 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4211677 0.81 KCNN4 (0.66) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL8653700 0.80 KCNN4 (0.60) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL4204126 0.78 KCNN4 (0.57) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL4211634 0.78 KCNN4 (0.57) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL11175731 0.77 ALDH1A1 (0.62) KCNN4ALDH1A1TSHRHTTNPSR1
SCHEMBL2005884 0.76 KCNN4 (0.56) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL4205517 0.76 KCNN4 (0.56) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL4207437 0.75 KCNN4 (0.55) KCNN4ALDH1A1TSHRHTTHPGD
SCHEMBL15542002 0.75 KCNN4 (1.00) KCNN4ALDH1A1
SCHEMBL4201420 0.74 KCNN4 (0.53) KCNN4ALDH1A1TSHRHTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019410-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 2000-07-19 EP disclosed
US-6060469-A Spiro-piperidine derivatives and their use as tachykinin antagonists MERCK SHARP & DOHME LTD. (GB) 2000-05-09 US disclosed
WO-1997019084-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1997-05-29 WO disclosed