SCHEMBL8112969

SCHEMBL8112969

COC(=O)c1ccc(CN(C(=O)C(c2ccccc2)c2ccccc2)[C@H](CCCNC(N)=N[N+](=O)[O-])C(N)=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.36
NPY1R P25929 1/20 0.35
NR3C1 P04150 1/20 0.34
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ROCK2 O75116 1/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
NPY4R P50391 1/20 0.32
LMNA P02545 1/20 0.32
MGLL Q99685 1/20 0.32
CCR5 P51681 1/20 0.32
CASR P41180 1/20 0.32
LPAR1 Q92633 1/20 0.32
LPAR5 Q9H1C0 1/20 0.32
F10 P00742 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8120178 0.92 NPY1R (0.36) F2NPY1RTMEM97SIGMAR1ALDH1A1
SCHEMBL8125838 0.92 NPY1R (0.35) F2NPY1RTMEM97SIGMAR1MAPT
SCHEMBL8119576 0.92 NPY1R (0.35) F2NPY1RTMEM97SIGMAR1MAPT
SCHEMBL8126826 0.91 CNR1 (0.37) F2NPY1RTMEM97SIGMAR1ALDH1A1
SCHEMBL7037398 0.90 MAPT (0.36) F2NPY1RALDH1A1MAPTHTT
SCHEMBL8121491 0.90 TMEM97 (0.37) F2NPY1RTMEM97SIGMAR1TDP1
SCHEMBL8119276 0.90 MEN1 (0.38) F2NPY1RMAPTHTTNPSR1
SCHEMBL8120508 0.89 F2 (0.38) F2NPY1RALDH1A1MAPTHTT
SCHEMBL8124247 0.89 NPY1R (0.42) F2NPY1RNPY4R
SCHEMBL8528491 0.89 NPY1R (0.35) F2NPY1RMAPTHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed