SCHEMBL8114282

SCHEMBL8114282

C[C@@H]1CNCCN1c1nc2ccccc2s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.46
NPC1 O15118 8/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
POLB P06746 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
TSHR P16473 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PPARG P37231 1/20 0.41
NCOA2 Q15596 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5342718 0.84 NPC1 (0.46) RAB9ANPC1SMN1; SMN2POLBCYP1A2
SCHEMBL19617714 0.82 NPC1 (0.53) RAB9ANPC1SMN1; SMN2MAPTLMNA
SCHEMBL10219276 0.82 NPC1 (0.52) RAB9ANPC1SMN1; SMN2POLBMAPT
SCHEMBL10219277 0.82 NPC1 (0.52) RAB9ANPC1SMN1; SMN2POLBMAPT
SCHEMBL10219282 0.82 NPC1 (0.52) RAB9ANPC1SMN1; SMN2POLBMAPT
SCHEMBL10219283 0.79 PPARD (0.51) CYP2D6PPARG
SCHEMBL10219278 0.79 PPARD (0.51) CYP2D6PPARG
SCHEMBL10219295 0.79 PPARD (0.51) CYP2D6PPARG
SCHEMBL9033466 0.79 RAB9A (0.49) RAB9ANPC1SMN1; SMN2POLBCYP1A2
SCHEMBL23744657 0.78 RAB9A (0.43) RAB9ANPC1SMN1; SMN2POLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed