SCHEMBL8116258

SCHEMBL8116258

CC(C)(C)C(O)C(C#N)c1ccc2ccccc2c1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 10/20 0.55
SLC6A4 P31645 10/20 0.55
SLC6A3 Q01959 10/20 0.55
UGT2B7 P16662 1/20 0.50
AOC3 Q16853 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ATM Q13315 1/20 0.44
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
KCNH2 Q12809 5/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3673974 0.83 UGT2B7 (0.56) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL5231024 0.82 UGT2B7 (0.53) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL8102026 0.80 TSHR (0.50) SLC6A2SLC6A4SLC6A3AOC3TSHR
SCHEMBL3663686 0.78 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3UGT2B7MEN1
SCHEMBL11547167 0.77 UGT2B7 (0.47) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL27469529 0.77 UGT2B7 (0.61) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL17455348 0.76 SLC6A2 (0.56) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL3041531 0.74 TSHR (0.57) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL27536762 0.74 TSHR (0.57) SLC6A2SLC6A4SLC6A3UGT2B7AOC3
SCHEMBL12004836 0.74 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3UGT2B7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069177-A ADMINISTERING TO THE HUMAN AN EFFECTIVE ANTIDEPRESSANT DOSE OF THE COMPOUND 3-HYDROXY-4,4-DIMETHYL-2-(2'-NAPHTHYL)PENTYL-N,N-DIMETHYLAMINE OR SALT THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (HK) 2000-05-30 US disclosed