SCHEMBL8117147

SCHEMBL8117147

CCOC(=O)c1cc(Br)cc(C)c1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.48
CA12 O43570 3/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA7 P43166 3/20 0.47
CA9 Q16790 3/20 0.47
CA14 Q9ULX7 3/20 0.47
TSHR P16473 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.44
CYP3A4 P08684 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 3/20 0.43
ALDH1A1 P00352 3/20 0.43
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
LMNA P02545 2/20 0.43
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179423 0.85 GAA (0.49) RXFP1CA12CA1CA2CA7
SCHEMBL10712967 0.83 CA12 (0.45) RXFP1CA12CA1CA2CA7
SCHEMBL3310733 0.82 KDR (0.43) CA12CA1CA2CA7CA9
SCHEMBL10627374 0.82 CA12 (0.59) CA12CA1CA2CA7CA9
SCHEMBL12326380 0.81 ALDH1A1 (0.47) CA12CA1CA2CA7CA9
SCHEMBL28532275 0.81 KDR (0.39) RXFP1SMN1; SMN2MAPTALDH1A1ALOX15
SCHEMBL4867955 0.79 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL17210813 0.79 KDM4E (0.44) RXFP1CA9CYP3A4MAPTALDH1A1
SCHEMBL27694753 0.79 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL2312711 0.79 MAPT (0.54) SMN1; SMN2TDP1MAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008147697-A1 BENZIMIDAZOLONE CHYMASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-12-04 WO disclosed