SCHEMBL8125656

SCHEMBL8125656

COc1ccc(-n2cnnn2)cc1C(C)=O

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
HPGD P15428 1/20 0.58
KCNJ1 P48048 2/20 0.57
KMT2A Q03164 4/20 0.52
TP53 P04637 1/20 0.52
PTGS2 P35354 2/20 0.52
PKM P14618 1/20 0.51
RXFP1 Q9HBX9 2/20 0.50
MEN1 O00255 2/20 0.50
EPHX2 P34913 1/20 0.49
TSHR P16473 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6425207 0.89 KMT2A (0.52) ALDH1A1HPGDKCNJ1KMT2ATP53
SCHEMBL6424185 0.88 TP53 (0.61) ALDH1A1HPGDKCNJ1KMT2ATP53
SCHEMBL6421265 0.88 KMT2A (0.51) ALDH1A1HPGDKCNJ1KMT2ATP53
SCHEMBL8130566 0.86 KMT2A (0.50) ALDH1A1HPGDKCNJ1KMT2ATP53
SCHEMBL8134305 0.85 TP53 (0.52) ALDH1A1HPGDKCNJ1KMT2ATP53
Iodomethane SCHEMBL8593226 0.83 TP53 (0.50) ALDH1A1HPGDKCNJ1KMT2ATP53
SCHEMBL12970651 0.81 RXFP1 (0.56) ALDH1A1HPGDKCNJ1KMT2ATP53
SCHEMBL8179017 0.77 ALDH1A1 (0.54) ALDH1A1HPGDKMT2ATP53PTGS2
SCHEMBL8530014 0.77 ALDH1A1 (0.54) ALDH1A1HPGDKMT2ATP53PTGS2
SCHEMBL8594200 0.76 ALDH1A1 (0.50) ALDH1A1HPGDKCNJ1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096766-A 3-benzylaminopiperidines as tachykinin receptor antagonists MERCK SHARP & DOHME LTD. (GB) 2000-08-01 US disclosed
EP-0866790-A1 3-BENZYLAMINOPYRROLIDINES AND -PIPERIDINES AS TACHYKININ RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1998-09-30 EP disclosed
WO-1997021702-A1 3-BENZYLAMINOPYRROLIDINES AND -PIPERIDINES AS TACHYKININ RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1997-06-19 WO disclosed