SCHEMBL8126286

SCHEMBL8126286

CC(C)(C)OC(=O)N1Cc2ccc(Oc3cccc(Cl)c3)cc2CC1C=O

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 7/20 0.49
GHSR Q92847 6/20 0.43
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
FFAR1 O14842 1/20 0.40
ADRB3 P13945 1/20 0.40
PTPN1 P18031 1/20 0.39
STS P08842 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12765134 0.87 HDAC8 (0.47) HDAC8GHSRMEN1KMT2AFFAR1
SCHEMBL1634598 0.86 HDAC8 (0.53) HDAC8PTPN1
SCHEMBL7945553 0.86 HDAC8 (0.53) HDAC8PTPN1
SCHEMBL1636444 0.84 PTPN1 (0.58) HDAC8PTPN1
SCHEMBL7935988 0.84 PTPN1 (0.58) HDAC8PTPN1
SCHEMBL29798802 0.81 HDAC8 (0.46) HDAC8MEN1KMT2APTPN1
SCHEMBL2730295 0.81 HDAC8 (0.46) HDAC8MEN1KMT2APTPN1
SCHEMBL19329217 0.78 HDAC8 (0.53) HDAC8PTPN1
SCHEMBL19329216 0.78 HDAC8 (0.53) HDAC8PTPN1
SCHEMBL8107263 0.78 ESR2 (0.64) HDAC8GHSRSTS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7829665-B2 Macrocyclic inhibitors of hepatitis C virus replication INTERMUNE, INC. (US) 2010-11-09 US disclosed
WO-2008141227-A1 NOVEL PEPTIDE INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2008-11-20 WO disclosed