SCHEMBL8126293

SCHEMBL8126293

COc1c(C(=O)NC2CC3CCCC(C2)N3Cc2ccccc2)cc(N)c2ccccc12

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.80
DRD2 P14416 2/20 0.69
DRD3 P35462 1/20 0.58
HTR3A P46098 1/20 0.58
OPRK1 P41145 2/20 0.56
CXCR6 O00574 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8125940 0.96 SIGMAR1 (0.74) SIGMAR1DRD2DRD3
SCHEMBL11890531 0.96 SIGMAR1 (0.74) SIGMAR1DRD2DRD3
SCHEMBL8124961 0.96 SIGMAR1 (0.74) SIGMAR1DRD2DRD3
SCHEMBL8118341 0.90 SIGMAR1 (0.65) SIGMAR1DRD2DRD3CXCR6
SCHEMBL8119845 0.89 SIGMAR1 (0.64) SIGMAR1DRD2DRD3
SCHEMBL8117971 0.89 SIGMAR1 (1.00) SIGMAR1DRD2DRD3
SCHEMBL8126235 0.86 SIGMAR1 (0.75) SIGMAR1DRD2DRD3CXCR6
SCHEMBL8127075 0.86 SIGMAR1 (0.75) SIGMAR1DRD2DRD3CXCR6
SCHEMBL8120009 0.86 SIGMAR1 (0.75) SIGMAR1DRD2DRD3
SCHEMBL8118831 0.86 SIGMAR1 (0.75) SIGMAR1DRD2DRD3HTR3AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861252-B1 NAPHTHAMIDE DERIVATIVES OF 3 BETA-AMINO AZABICYCLO OCTANE OR NONANE AS NEUROLEPTIC AGENTS PF MEDICAMENT (FR) 2000-02-23 EP claimed