SCHEMBL8128283

SCHEMBL8128283

COc1ccc2c(c1)c(C1=C(c3cn(CC(C)N(C)C)c4ccccc34)C(=O)NC1=O)cn2C

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 4/20 0.61
GSK3B P49841 4/20 0.61
PRKD1 Q15139 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
CCNE2 O96020 2/20 0.57
CDK4 P11802 2/20 0.57
CCND1 P24385 2/20 0.57
CCNE1 P24864 2/20 0.57
CDK2 P24941 2/20 0.57
PIM1 P11309 1/20 0.56
PRKACA P17612 1/20 0.56
PRKACG P22612 1/20 0.56
PRKACB P22694 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8161651 0.85 GSK3B (0.80) PRKCAGSK3BCCNE2CDK4CCND1
SCHEMBL8120702 0.84 PRKCA (0.80) PRKCAGSK3BPRKD1TDP1CCNE2
SCHEMBL14041601 0.82 GSK3B (0.66) PRKCAGSK3BPIM1PRKACAPRKACG
SCHEMBL30834694 0.82 PRKCA (0.64) PRKCAGSK3BCCNE2CDK4CCND1
SCHEMBL8122419 0.82 CCNT1 (0.66) PRKCAGSK3BPRKD1TDP1CDK2
SCHEMBL8127999 0.82 CCNT1 (0.66) PRKCAGSK3BPRKD1TDP1CDK2
SCHEMBL8122774 0.81 PRKCA (0.63) PRKCAGSK3BPRKD1TDP1CDK2
SCHEMBL8113347 0.81 PRKCA (0.63) PRKCAGSK3BPRKD1TDP1CDK2
SCHEMBL8075384 0.80 PRKCA (0.61) PRKCAGSK3BPIM1
SCHEMBL7502631 0.80 GSK3B (0.70) PRKCAGSK3BCCNE2CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0642513-B1 INDOLOCARBAZOLE IMIDES AND THEIR USE KTB TUMORFORSCHUNGSGESELLSCHAF (DE) 2000-08-09 EP disclosed
EP-0642513-A1 INDOLOCARBAZOLE IMIDES AND THEIR USE GÖDECKE AKTIENGESELLSCHAFT (DE) 1995-03-15 EP disclosed
WO-1993024491-A1 INDOLOCARBAZOLE IMIDES AND THEIR USE Gödecke Aktiengesellschaft (DE) 1993-12-09 WO disclosed