SCHEMBL8128993

SCHEMBL8128993

O=C(C=CC1CCN(Cc2cccs2)CC1)c1ccc(Nc2ncnc3c2CCC3)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.35
EGFR P00533 2/20 0.35
KDR P35968 1/20 0.35
PYGM P11217 4/20 0.34
HDAC8 Q9BY41 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CXCR3 P49682 1/20 0.33
PARP1 P09874 1/20 0.33
SMARCA4 P51532 1/20 0.33
PBRM1 Q86U86 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
LTA4H P09960 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128991 1.00 TRPV1 (0.35) TRPV1EGFRKDRPYGMHDAC8
SCHEMBL8126483 0.87 HDAC8 (0.48) HDAC8HDAC6KDM4EALDH1A1MAPT
SCHEMBL8126478 0.87 HDAC8 (0.48) HDAC8HDAC6KDM4EALDH1A1MAPT
SCHEMBL8133214 0.85 HDAC8 (0.48) HDAC8HDAC6KDM4EALDH1A1MAPT
SCHEMBL8133217 0.85 HDAC8 (0.48) HDAC8HDAC6KDM4EALDH1A1MAPT
SCHEMBL8125056 0.84 HTR2A (0.41) HDAC8SIGMAR1HDAC6
SCHEMBL8125059 0.84 HTR2A (0.41) HDAC8SIGMAR1HDAC6
SCHEMBL8922063 0.83 ACHE (0.41) TRPV1LTA4HEPHX2
SCHEMBL8133359 0.83 HDAC8 (0.40) EGFRHDAC8SIGMAR1
SCHEMBL8133357 0.83 HDAC8 (0.40) EGFRHDAC8SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664291-B1 PYRIMIDINE COMPOUND UBE INDUSTRIES (JP) 2000-07-19 EP disclosed
US-5610303-A MONOAMIDE OXIDASE INHIBITORS UBE INDUSTRIES, LTD. (JP) 1997-03-11 US disclosed
EP-0664291-A1 PYRIMIDINE COMPOUND UBE INDUSTRIES, LTD. (JP) 1995-07-26 EP disclosed