SCHEMBL8129015

SCHEMBL8129015

Fc1c[c]c(Oc2cccc(Cl)c2Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.43
SLC6A2 P23975 10/20 0.43
SLC6A4 P31645 4/20 0.43
SLC6A3 Q01959 3/20 0.43
ALDH1A1 P00352 3/20 0.40
RHEB Q15382 1/20 0.40
NPSR1 Q6W5P4 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
ATM Q13315 1/20 0.33
SLC22A12 Q96S37 1/20 0.32
MEN1 O00255 1/20 0.32
TTR P02766 1/20 0.32
HSP90AA1 P07900 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
HSPB1 P04792 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8125202 0.85 ALDH1A1 (0.41) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8123023 0.82 ALDH1A1 (0.39) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8125043 0.82 ALDH1A1 (0.39) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8123025 0.81 KMT2A (0.43) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8125381 0.81 ALDH1A1 (0.38) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8130154 0.80 CASR (0.38) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8122855 0.79 SLC6A2 (0.35) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8115497 0.78 AR (0.38) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8127275 0.78 ALDH1A1 (0.41) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8131299 0.78 SLC6A2 (0.41) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028945-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS Amgen Inc. (US) 2000-08-23 EP disclosed
WO-1999024404-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC. (US) 1999-05-20 WO disclosed