SCHEMBL8129146

SCHEMBL8129146

Cc1ccccc1[C@H](Br)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 1/20 0.46
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
ESR1 P03372 1/20 0.43
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 1/20 0.40
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP2D6 P10635 1/20 0.37
SRC P12931 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CTSA P10619 1/20 0.36
HPGD P15428 2/20 0.36
MYC P01106 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL76634 1.00 ACP3 (0.46) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL5925059 1.00 ACP3 (0.46) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL9278678 0.83 ESR1 (0.43) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL9276808 0.82 HSP90AA1 (0.44) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL8763320 0.82 ALDH1A1 (0.46) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL5389348 0.82 CYP1A2 (0.54) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL9127138 0.79 KMT2A (0.44) ACP3ESR1ALDH1A1MEN1KMT2A
SCHEMBL5618977 0.79 ESR1 (0.39) ACP3CES2CES1ESR1ALDH1A1
SCHEMBL4370114 0.78 ACP3 (0.48) ACP3ESR1ALDH1A1LMNAL3MBTL1
SCHEMBL2206363 0.78 SRC (0.50) ACP3ESR1ALDH1A1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124343-A Substituted phenyl compounds with a substituent having a thienyl ring RHONE-POULENC RORER LIMITED (GB) 2000-09-26 US disclosed
EP-0805802-B1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LTD (GB) 2000-08-16 EP disclosed
US-6048893-A Substituted phenyl compounds with a substituent having A 1,3-benzodioxole ring RHONE-POULENC RORER LIMITED (GB) 2000-04-11 US disclosed
EP-0805802-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE-POULENC RORER LIMITED (GB) 1997-11-12 EP disclosed
WO-1996022978-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LIMITED (GB) 1996-08-01 WO disclosed