SCHEMBL8129242

SCHEMBL8129242

O=C(O)Oc1cn(C2CC2)c2c(F)c(N3CCC(N=Cc4ccc([N+](=O)[O-])cc4)C3)c(F)cc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 4/20 0.41
TOP1 P11387 2/20 0.41
KCNH2 Q12809 4/20 0.40
ALDH1A1 P00352 3/20 0.40
POLB P06746 2/20 0.40
OPRM1 P35372 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
OPRD1 P41143 1/20 0.40
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
PRKD3 O94806 1/20 0.39
ALOX15 P16050 1/20 0.39
CLK2 P49760 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
BCHE P06276 2/20 0.39
ACHE P22303 2/20 0.39
BACE1 P56817 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8120307 0.92 TOP2A (0.40) TOP2ATOP1KCNH2ALDH1A1POLB
SCHEMBL8134768 0.91 KCNH2 (0.43) TOP2AKCNH2ALDH1A1POLBOPRM1
SCHEMBL8119666 0.91 KCNH2 (0.43) TOP2AKCNH2ALDH1A1POLBOPRM1
SCHEMBL8901293 0.90 ALDH1A1 (0.51) TOP2ATOP1KCNH2ALDH1A1POLB
SCHEMBL8565145 0.90 ALDH1A1 (0.51) TOP2ATOP1KCNH2ALDH1A1POLB
SCHEMBL8901278 0.90 ALDH1A1 (0.51) TOP2ATOP1KCNH2ALDH1A1POLB
SCHEMBL8122322 0.90 KCNH2 (0.45) TOP2AKCNH2ALDH1A1POLBOPRM1
SCHEMBL8136563 0.88 KCNH2 (0.43) TOP2AKCNH2ALDH1A1POLBOPRM1
SCHEMBL8138031 0.87 KCNH2 (0.40) TOP2ATOP1KCNH2ALDH1A1POLB
SCHEMBL8129317 0.85 ALDH1A1 (0.48) TOP2ATOP1KCNH2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0401623-B1 Process for the preparation of 7-(3-amino- and 3-aminomethyl-1-pyrrolidinyl)-3-quinolinonecarboxylic and -naphthyridinonecarboxylic acids BAYER AG (DE) 2000-01-26 EP disclosed
EP-0401623-A1 Process for the preparation of 7-(3-amino- and 3-aminomethyl-1-pyrrolidinyl)-3-quinolinonecarboxylic and -naphthyridinonecarboxylic acids BAYER AG (DE) 1990-12-12 EP disclosed