SCHEMBL8133136

SCHEMBL8133136

Cc1oc(-c2ccccc2)nc1CCOc1ccc(/C=C2\SC(=O)NC2=O)cn1

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PPARG P37231 20/20 0.57
PPARA Q07869 19/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8133138 1.00 PPARG (0.57) PPARGPPARA
SCHEMBL8141923 0.91 KCNH2 (0.50) PPARGPPARA
SCHEMBL8141922 0.91 KCNH2 (0.50) PPARGPPARA
SCHEMBL10366704 0.90 HPGD (0.61) PPARGPPARA
SCHEMBL10364994 0.90 HPGD (0.61) PPARGPPARA
SCHEMBL10364971 0.90 HPGD (0.61) PPARGPPARA
SCHEMBL8133143 0.89 PPARG (0.55) PPARGPPARA
SCHEMBL6966781 0.83 PPARG (0.52) PPARGPPARA
SCHEMBL6966778 0.83 PPARG (0.52) PPARGPPARA
SCHEMBL9316520 0.82 PIM1 (0.45) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0605228-A1 Thiazolidinedione derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-07-06 EP claimed
EP-0605228-B1 Thiazolidinedione derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-03-01 EP disclosed
US-5489602-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-02-06 US disclosed
EP-0605228-A1 Thiazolidinedione derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-07-06 EP disclosed