SCHEMBL8133207

SCHEMBL8133207

CC(C)[C@H](N)C(=O)NN1C(=O)C(CC2CC2)c2ccccc2-c2ccccc21.CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)NN1C(=O)C(CC2CC2)c2ccccc2-c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ATM Q13315 1/20 0.40
SCN9A Q15858 12/20 0.37
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
CA2 P00918 1/20 0.36
CASP3 P42574 1/20 0.34
CCKAR P32238 1/20 0.34
CCKBR P32239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307634 0.95 KMT2A (0.42) KMT2AMEN1ATMSCN9APSEN1
SCHEMBL6313103 0.88 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6306703 0.87 KMT2A (0.41) KMT2AATMSCN9APSEN1PSEN2
Hydrochloric Acid SCHEMBL4413424 0.87 PSEN1 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8140471 0.82 CA2 (0.38) KMT2AMEN1ATMSCN9APSEN1
SCHEMBL6309257 0.81 MEN1 (0.37) KMT2AMEN1ATMSCN9APSEN1
SCHEMBL6308554 0.81 PSEN1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7568374 0.81 SCN9A (0.39) KMT2AMEN1ATMSCN9APSEN1
SCHEMBL4418511 0.81 SCN9A (0.39) KMT2AMEN1ATMSCN9APSEN1
SCHEMBL4424746 0.81 SCN9A (0.39) KMT2AMEN1ATMSCN9APSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042298-A1 POLYCYCLIC ALPHA-AMINO-EPSILON-CAPROLACTAMS AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2000-10-11 EP claimed
WO-1999032453-A1 POLYCYCLIC α-AMINO-⊂-CAPROLACTAMS AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 1999-07-01 WO claimed