SCHEMBL8134677

SCHEMBL8134677

CN(c1cncn1Cc1ccc(S(C)(=O)=O)cc1)C1CCOc2c(C(=O)N[C@@H](Cc3ccc(Cl)cc3)C(N)=O)cccc21

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.33
ITGA4 P13612 4/20 0.33
ITGB7 P26010 2/20 0.33
BCL2 P10415 3/20 0.33
BCL2L1 Q07817 2/20 0.33
MCL1 Q07820 2/20 0.33
CAPN1 P07384 2/20 0.32
CTSB P07858 2/20 0.32
MC4R P32245 3/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
CA2 P00918 1/20 0.32
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA9 Q16790 2/20 0.31
P2RX3 P56373 1/20 0.31
KCNA5 P22460 1/20 0.31
CCR1 P32246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128898 0.93 CAPN1 (0.39) BCL2BCL2L1MCL1CAPN1CTSB
SCHEMBL8143718 0.91 P2RX3 (0.35) ITGB1CAPN1CTSBP2RX3
SCHEMBL8125473 0.90 CCR3 (0.38) BCL2BCL2L1MCL1CAPN1CTSB
SCHEMBL8134169 0.90 P2RX3 (0.35) BCL2CAPN1CTSBP2RX3
SCHEMBL8133580 0.90 FNTA (0.37)
SCHEMBL8141784 0.87 CAPN1 (0.36) ITGB1ITGA4ITGB7CAPN1CTSB
SCHEMBL8135109 0.85 P2RX3 (0.34) P2RX3KCNA5
SCHEMBL8134680 0.85 FNTA (0.37) ITGB1ITGA4ITGB7
SCHEMBL8134674 0.85 FNTA (0.37) ITGB1ITGA4ITGB7
SCHEMBL8140831 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054882-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 2000-11-29 EP disclosed
WO-1999041248-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AVENTIS PHARMA S.A. (FR) 1999-08-19 WO disclosed