SCHEMBL8137019

SCHEMBL8137019

CSc1nc(SCc2ccccn2)nc(Cl)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 4/20 0.42
RAB9A P51151 6/20 0.40
NPC1 O15118 5/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 4/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 3/20 0.39
CYP2E1 P05181 2/20 0.39
CYP2C8 P10632 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2B6 P20813 2/20 0.39
CYP2C19 P33261 2/20 0.39
KDM4E B2RXH2 2/20 0.38
TSHR P16473 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637738 0.88 METAP2 (0.48) METAP2RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL8134818 0.85 SMN1; SMN2 (0.40) METAP2RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL6636431 0.82 METAP2 (0.44) METAP2RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL8125882 0.76 HTT (0.39) RAB9ANPC1SMN1; SMN2LMNAMAPT
SCHEMBL8140855 0.75 SMN1; SMN2 (0.41) METAP2RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL6639693 0.74 NPC1 (0.47) METAP2RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL6638720 0.72 METAP2 (0.44) METAP2RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL6639863 0.70 NPC1 (0.61) METAP2RAB9ANPC1SMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL10560721 0.69 NPC1 (0.51) METAP2RAB9ANPC1SMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL10562402 0.69 NPC1 (0.59) METAP2RAB9ANPC1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124306-A Thioalkyl alpha substituted pyrimidine compounds PHARMACIA & UPJOHN COMPANY (US) 2000-09-26 US disclosed
EP-1034167-A1 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 2000-09-13 EP disclosed
WO-1999019304-A9 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS UPJOHN CO (US) 1999-07-08 WO disclosed
WO-1999019304-A2 ALPHA-ALKYLTHIO SUBSTITUTED PYRIMIDINE ETHERS AND THIOETHERS AS VIRAL REVERSE TRANSCRIPTASE INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1999-04-22 WO disclosed