SCHEMBL8137183

SCHEMBL8137183

Nc1cccc(-c2c[nH]cn2)c1N

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.33
CD44 P16070 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
PARP1 P09874 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ADORA3 P0DMS8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1501942 0.85 IDO1 (0.47) IDO1ALDH1A1L3MBTL1DCUN1D1KDM4E
Hydrochloric Acid SCHEMBL1502211 0.83 IDO1 (0.46) IDO1ALDH1A1L3MBTL1DCUN1D1KDM4E
Hydrochloric Acid SCHEMBL1502209 0.83 IDO1 (0.46) IDO1ALDH1A1L3MBTL1DCUN1D1KDM4E
SCHEMBL26259557 0.78 IKBKE (0.32) PARP1
SCHEMBL26259713 0.73 ALDH1A1 (0.43) ALDH1A1L3MBTL1PARP1KDM4EGAA
SCHEMBL27958628 0.70 CDK2 (0.39) IDO1DCUN1D1PARP1NPC1
SCHEMBL26259238 0.70 NISCH (0.41) ALDH1A1KDM4ENPC1GAAHSD17B10
SCHEMBL26259398 0.70 MEN1 (0.33) PARP1
SCHEMBL560128 0.70 ALDH1A1 (0.56) CD44ALDH1A1L3MBTL1PARP1HSD17B10
SCHEMBL16147908 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0556393-B1 FUSED PYRAZINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 2000-07-26 EP disclosed
US-5283244-A Anticonvulsants, nervous system disorders YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-02-01 US disclosed
EP-0556393-A1 FUSED PYRAZINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1993-08-25 EP disclosed