SCHEMBL8137273

SCHEMBL8137273

CCOC(=O)c1ccc2c(c1OC)C(=O)C(C)(C)CS2(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
KDM4E B2RXH2 4/20 0.35
HSD17B10 Q99714 3/20 0.35
CA12 O43570 2/20 0.35
CA2 P00918 2/20 0.35
CA7 P43166 2/20 0.35
CA9 Q16790 2/20 0.35
CA14 Q9ULX7 2/20 0.35
CA1 P00915 1/20 0.35
ALDH1A1 P00352 5/20 0.34
MAPK1 P28482 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
NPC1 O15118 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7134324 0.70 TSHR (0.41) TSHRKDM4EHSD17B10CA12CA2
SCHEMBL7134321 0.69 CA12 (0.43) TSHRKDM4EHSD17B10CA12CA2
SCHEMBL8134865 0.68 PDK2 (0.35) TSHRKDM4EHSD17B10ALDH1A1KMT2A
SCHEMBL8136245 0.67 TSHR (0.38) TSHRKDM4EHSD17B10CA12CA2
SCHEMBL7890058 0.66 TSHR (0.40) TSHRKDM4EHSD17B10CA12CA2
SCHEMBL23773427 0.66 TSHR (0.68) TSHRKDM4EHSD17B10CA12CA2
SCHEMBL6613660 0.65 KMT2A (0.59) TSHRCA12CA2CA7CA9
SCHEMBL7131946 0.65 ALDH1A1 (0.39) TSHRKDM4EHSD17B10ALDH1A1MAPK1
SCHEMBL28750763 0.64 ALDH1A1 (0.51) TSHRKDM4EHSD17B10CA12CA2
SCHEMBL11678098 0.63 TSHR (0.63) TSHRKDM4EHSD17B10CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6159904-A Pyrazole derivatives IDEMITSU KOSAN CO., LTD. (JP) 2000-12-12 US disclosed
EP-0970956-A1 PYRAZOLE DERIVATIVES IDEMITSU KOSAN COMPANY LIMITED (JP) 2000-01-12 EP disclosed