SCHEMBL8137992

SCHEMBL8137992

CN1CCN(c2cc3c(cc2Br)CCN3C(=O)Nc2cccc3c(-c4ccncc4)cccc23)CC1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.72
HTR1D P28221 4/20 0.72
HTR1B P28222 4/20 0.72
SLC2A1 P11166 2/20 0.53
HTR2B P41595 4/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
NFKB1 P19838 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
HTR2C P28335 10/20 0.44
HTR2A P28223 8/20 0.44
WDR5 P61964 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8127323 0.95 HTR1A (0.81) HTR1AHTR1DHTR1BSLC2A1HTR2B
SCHEMBL8122308 0.90 HTR1A (0.73) HTR1AHTR1DHTR1BSLC2A1HTR2C
SCHEMBL8143058 0.89 HTR1D (0.90) HTR1AHTR1DHTR1BSLC2A1HTR2B
SCHEMBL8125735 0.89 HTR1D (0.57) HTR1AHTR1DHTR1BSLC2A1HTR2B
SCHEMBL8128398 0.88 HTR1D (0.70) HTR1AHTR1DHTR1BHTR2BCYP1A2
SCHEMBL8196349 0.86 HTR1A (0.56) HTR1AHTR1DHTR1BSLC2A1HTR2C
SCHEMBL8119474 0.85 HTR1A (0.82) HTR1AHTR1DHTR1BSLC2A1HTR2B
SCHEMBL8130546 0.84 HTR1A (0.57) HTR1AHTR1DHTR1BSLC2A1HTR2B
SCHEMBL8121210 0.84 HTR1A (1.00) HTR1AHTR1DHTR1BSLC2A1HTR2B
SCHEMBL8128007 0.83 HTR1A (0.79) HTR1AHTR1DHTR1BSLC2A1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975593-A1 INDOLE DERIVATIVES HAVING COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2000-02-02 EP disclosed
WO-1998050358-A1 INDOLE DERIVATIVES HAVING COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed