SCHEMBL8140959

SCHEMBL8140959

Nc1ccc(Cn2cncc2C=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 14/20 0.67
CYP11B2 P19099 14/20 0.67
IDO1 P14902 1/20 0.38
CYP19A1 P11511 2/20 0.38
HTR6 P50406 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
CYP17A1 P05093 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758083 0.85 CYP11B1 (0.68) CYP11B1CYP11B2IDO1CYP19A1ALDH1A1
SCHEMBL7986619 0.84 CYP11B1 (0.67) CYP11B1CYP11B2IDO1CYP19A1
SCHEMBL765399 0.84 CYP11B1 (0.67) CYP11B1CYP11B2IDO1CYP19A1ALDH1A1
SCHEMBL7696780 0.84 CYP11B1 (0.67) CYP11B1CYP11B2IDO1CYP19A1ALDH1A1
SCHEMBL7700254 0.84 CYP11B1 (0.67) CYP11B1CYP11B2IDO1CYP19A1ALDH1A1
SCHEMBL7696643 0.83 CYP11B1 (0.66) CYP11B1CYP11B2IDO1CYP19A1ALDH1A1
SCHEMBL1757759 0.83 CYP11B1 (0.66) CYP11B1CYP11B2IDO1CYP19A1ALDH1A1
SCHEMBL8135755 0.83 CYP11B1 (0.65) CYP11B1CYP11B2IDO1ALDH1A1
SCHEMBL5935193 0.81 CYP11B1 (0.63) CYP11B1CYP11B2IDO1CYP19A1FNTA
SCHEMBL8133106 0.81 CYP11B1 (0.63) CYP11B1CYP11B2IDO1CYP19A1FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054882-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 2000-11-29 EP disclosed
WO-1999041248-A1 CONDENSED HETEROCYCLIC SYSTEM DERIVATIVES, PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AVENTIS PHARMA S.A. (FR) 1999-08-19 WO disclosed