SCHEMBL8142196

SCHEMBL8142196

O=C(O)/C=C1/c2ccccc2COc2cc(CCl)ccc21

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.53
HRH1 P35367 3/20 0.46
LMNA P02545 1/20 0.43
TBXA2R P21731 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8142200 1.00 AKR1B1 (0.53) AKR1B1HRH1LMNATBXA2R
SCHEMBL8137781 0.89 AKR1B1 (0.54) AKR1B1HRH1LMNATBXA2R
SCHEMBL8137785 0.89 AKR1B1 (0.54) AKR1B1HRH1LMNATBXA2R
SCHEMBL8614712 0.81 HRH1 (0.50) HRH1LMNA
SCHEMBL8614715 0.81 HRH1 (0.50) HRH1LMNA
SCHEMBL8143124 0.81 TBXA2R (0.53) TBXA2R
SCHEMBL8143121 0.81 TBXA2R (0.53) TBXA2R
SCHEMBL8126089 0.79 AKR1B1 (0.43) AKR1B1HRH1LMNA
SCHEMBL8126092 0.79 AKR1B1 (0.43) AKR1B1HRH1LMNA
SCHEMBL9045798 0.73 TBXA2R (0.58) TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549352-B1 Tricyclic compounds as angiotensin II antagonists KYOWA HAKKO KOGYO KK (JP) 2000-03-01 EP disclosed
US-5478840-A Imidazo(4,5-b)pyridine derivatives used as antagonism to angiotensin ii receptors KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-12-26 US disclosed
US-5378701-A Angiotensin II inhibitors; hypotensive agents; congestive heart and kidney failure; glaucoma KYOWA HAKKO KOGYO (JP) 1995-01-03 US disclosed
EP-0549352-A2 Tricyclic compounds as angiotensin II antagonists KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-06-30 EP disclosed