SCHEMBL8142359

SCHEMBL8142359

Cc1nc2c([nH]1)c(=O)[nH]c(=O)n2Cc1ccco1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
LMNA P02545 1/20 0.67
CYP1A1 P04798 1/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
NFKB1 P19838 1/20 0.67
MAPK1 P28482 1/20 0.67
CYP2C19 P33261 1/20 0.67
BLM P54132 1/20 0.67
PMP22 Q01453 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
HIF1A Q16665 1/20 0.67
TSHR P16473 4/20 0.51
PNP P00491 2/20 0.51
ADORA2B P29275 6/20 0.51
ADORA2A P29274 5/20 0.51
ALDH1A1 P00352 3/20 0.47
POLB P06746 2/20 0.46
PKM P14618 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Furafylline SCHEMBL191214 0.81 MEN1 (1.00) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL4624542 0.80 PNP (0.60) MEN1KMT2ABLMTSHRPNP
SCHEMBL6346663 0.74 ADORA2A (0.59) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL10963141 0.73 ADORA2A (0.55) MEN1KMT2ALMNABLMSMN1; SMN2
SCHEMBL8128166 0.72 MEN1 (0.67) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL8143264 0.72 MEN1 (0.67) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL8128164 0.72 MEN1 (0.67) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL8135676 0.70 TSHR (0.62) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL10979332 0.70 ADORA2A (0.41) MEN1KMT2ALMNACYP1A1CYP1A2
SCHEMBL5646 0.70 PDE2A (0.61) MEN1KMT2ALMNAMAPK1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6075029-A Xanthine modulators of metabolism of cellular P-450 CELL THERAPEUTICS, INC. (US) 2000-06-13 US disclosed