SCHEMBL8135676

SCHEMBL8135676

Nc1c(N)n(Cc2ccco2)c(=O)[nH]c1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.62
MEN1 O00255 8/20 0.51
KMT2A Q03164 8/20 0.51
ALDH1A1 P00352 6/20 0.51
PKM P14618 4/20 0.51
MAPT P10636 4/20 0.51
POLB P06746 4/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
PNP P00491 2/20 0.51
HSD17B10 Q99714 2/20 0.51
HPGD P15428 2/20 0.51
APEX1 P27695 2/20 0.47
RECQL P46063 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
BLM P54132 2/20 0.47
KDM4E B2RXH2 1/20 0.47
UHRF1 Q96T88 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.47
GAA P10253 1/20 0.46
MAPK1 P28482 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1958885 0.86 TSHR (0.52) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL2557771 0.83 TSHR (0.56) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL8133362 0.77 TSHR (1.00) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL1945491 0.76 KDM4E (0.66) TSHRMEN1KMT2AALDH1A1MAPT
SCHEMBL11362739 0.74 TSHR (0.59) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL1960199 0.70 ALDH1A1 (0.49) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL8142359 0.70 MEN1 (0.67) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL6346663 0.70 ADORA2A (0.59) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL2588131 0.70 TSHR (1.00) TSHRMEN1KMT2AALDH1A1PKM
SCHEMBL1944329 0.70 TLR7 (0.49) MEN1KMT2AALDH1A1PKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6075029-A Xanthine modulators of metabolism of cellular P-450 CELL THERAPEUTICS, INC. (US) 2000-06-13 US disclosed
WO-1999035148-A1 COMPOUNDS FOR INCREASED BIOAVAILABILITY CELL THERAPEUTICS, INC. (US) 1999-07-15 WO disclosed