SCHEMBL8143249

SCHEMBL8143249

O=C(O)CN1C(=O)C(=O)N(Cc2ccccc2Cl)C1=O

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C19 P33261 1/20 0.61
KMT2A Q03164 3/20 0.54
NLRP3 Q96P20 1/20 0.52
MEN1 O00255 1/20 0.52
CTDSP1 Q9GZU7 1/20 0.52
CA12 O43570 1/20 0.47
CA9 Q16790 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8151552 0.85 CYP1A2 (0.51) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL23440033 0.84 F2 (0.60) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL8144393 0.82 PTPN1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL8143584 0.82 KMT2A (0.76) CYP2D6CYP2C19KMT2ACA12CA9
SCHEMBL8143252 0.82 KMT2A (0.53) KMT2AMEN1CA12CA9MAPT
SCHEMBL9323617 0.81 KMT2A (0.73) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL8871694 0.80 KMT2A (0.46) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL6967373 0.79 TDP1 (0.51) CYP1A2KMT2AMEN1CA12CA9
SCHEMBL8872105 0.78 KMT2A (0.47) KMT2AMEN1CA12CA9
SCHEMBL8134728 0.78 USP2 (0.52) CYP1A2CYP3A4CYP2C19KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6040326-A 3-deoxyglucosone production inhibitor NIPPON ZOKI PHARMACEUTICALS CO., LTD. (JP) 2000-03-21 US disclosed
EP-0855182-A1 3-Deoxyglucosone production inhibitor NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1998-07-29 EP disclosed
EP-0353198-B1 Parabanic acid derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO (JP) 1994-02-02 EP disclosed
US-4985453-A DIABETES TREATMENT NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1991-01-15 US disclosed
EP-0353198-A1 Parabanic acid derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1990-01-31 EP disclosed