SCHEMBL8144341

SCHEMBL8144341

CC(=O)NCC(=O)N1CCN(CC2CCN(C)CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.53
CACNA1B Q00975 2/20 0.53
CACNB1 Q02641 2/20 0.53
CACNA1C Q13936 1/20 0.53
FAP Q12884 2/20 0.40
DPP4 P27487 1/20 0.40
PREP P48147 1/20 0.40
BDKRB1 P46663 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GNAI3 P08754 1/20 0.38
GNAO1 P09471 1/20 0.38
GNAI1 P63096 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
KDM1A O60341 2/20 0.36
MAOB P27338 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23173625 0.94 CACNA2D1 (0.47) CACNA2D1CACNA1BCACNB1CACNA1CFAP
SCHEMBL23173789 0.87 CACNA2D1 (0.41) CACNA2D1CACNA1BCACNB1CACNA1CFAP
SCHEMBL24307350 0.86 CACNA2D1 (0.51) CACNA2D1CACNA1BCACNB1CACNA1CBDKRB1
SCHEMBL25571572 0.85 CACNA2D1 (0.55) CACNA2D1CACNA1BCACNB1CACNA1CBDKRB1
SCHEMBL1308937 0.82 MEN1 (0.54) CACNA2D1CACNA1BCACNB1CACNA1CBDKRB1
SCHEMBL8230809 0.81 TDP1 (0.50) FAPDPP4PREPNPSR1L3MBTL1
SCHEMBL8138867 0.81 CACNA2D1 (0.44) CACNA2D1CACNA1BCACNB1CACNA1CNPSR1
SCHEMBL23174010 0.81 CACNA2D1 (0.45) CACNA2D1CACNA1BCACNB1CACNA1CBDKRB1
SCHEMBL4067141 0.80 CYP1A2 (0.55) CACNA2D1CACNA1BCACNB1CACNA1CBDKRB1
SCHEMBL26705105 0.79 CACNA2D1 (0.49) CACNA2D1CACNA1BCACNB1CACNA1CBDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008119741-A2 3-IMIDAZOLYL-INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISEASES NOVARTIS AG (CH) 2008-10-09 WO disclosed