SCHEMBL8147229

SCHEMBL8147229

CN1C[C@@H]2CCc3[nH]c4ccc(Br)cc4c3[C@@H]2C1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.42
BAZ2B Q9UIF8 2/20 0.39
DHODH Q02127 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MCHR1 Q99705 4/20 0.38
MAPKAPK2 P49137 1/20 0.38
CYP2D6 P10635 2/20 0.36
KCNH2 Q12809 1/20 0.36
AXL P30530 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154453 0.82 MCHR1 (0.49) MCHR1CYP2D6KCNH2
SCHEMBL8154457 0.82 MCHR1 (0.49) MCHR1CYP2D6KCNH2
SCHEMBL782565 0.82 MCHR1 (0.49) MCHR1CYP2D6KCNH2
SCHEMBL8141837 0.82 MAPT (0.31) MAPTHRH3
Fumaric Acid SCHEMBL8146701 0.73 KMT2A (0.43) MCHR1KCNH2
Fumaric Acid SCHEMBL8155294 0.70 HRH4 (0.40) MAPTBAZ2BMCHR1KCNH2HRH3
Fumaric Acid SCHEMBL8373626 0.70 HRH4 (0.40) MAPTBAZ2BMCHR1KCNH2HRH3
SCHEMBL8372824 0.70 MCHR1 (0.38) MAPTHSD17B10MCHR1
SCHEMBL1988850 0.68 SIGMAR1 (0.67)
SCHEMBL12868041 0.65 BAZ2B (0.56) MAPTBAZ2BHSD17B10CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6063803-A ANALGESICS AND CHEMICAL INTERMEDIATES ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-05-16 US disclosed