SCHEMBL8147369

SCHEMBL8147369

[C-]#[N+]c1cc2ccc(Br)cc2cc1C

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
NCEH1 Q6PIU2 1/20 0.33
BACE1 P56817 1/20 0.32
DHODH Q02127 1/20 0.31
LMNA P02545 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8150148 1.00 CYP2A6 (0.42) CYP2A6KDM4EMEN1ALDH1A1MAPT
SCHEMBL8149480 0.80
SCHEMBL8404534 0.80 CYP2A6 (0.56) CYP2A6KDM4EMEN1ALDH1A1MAPT
SCHEMBL12126083 0.78 ALDH1A1 (0.35) CYP2A6ALDH1A1
SCHEMBL8140915 0.78 CYP2A6 (0.39) CYP2A6MEN1ALDH1A1KMT2A
SCHEMBL324210 0.78 ALDH1A1 (0.35) CYP2A6MEN1ALDH1A1MAPTKMT2A
SCHEMBL29955874 0.78 ALDH1A1 (0.35) CYP2A6MEN1ALDH1A1MAPTKMT2A
SCHEMBL8154003 0.78 CYP2A6 (0.42) CYP2A6ALDH1A1
SCHEMBL8155348 0.78 CYP1A2 (0.42) CYP2A6BACE1
SCHEMBL8150150 0.78 CYP2A6 (0.42) CYP2A6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116399-A1 Inhibitors of factor Xa MILLENNIUM PHARMACEUTICALS, INC. 2004-06-17 US disclosed