SCHEMBL8147403

SCHEMBL8147403

COc1ccccc1Nc1cc2n(c(=O)n1)CCc1ccccc1-2

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.71
MEN1 O00255 4/20 0.71
ATM Q13315 1/20 0.71
POLB P06746 5/20 0.70
KDM4E B2RXH2 10/20 0.64
PDE4A P27815 1/20 0.56
GPR84 Q9NQS5 1/20 0.56
ALDH1A1 P00352 8/20 0.55
HPGD P15428 5/20 0.55
MAPT P10636 4/20 0.55
HTT P42858 2/20 0.55
RXFP1 Q9HBX9 1/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
CASP6 P55212 1/20 0.54
CACNA1B Q00975 1/20 0.54
APBA1 Q02410 1/20 0.54
SIRT5 Q9NXA8 1/20 0.54
HSD17B10 Q99714 7/20 0.53
TSHR P16473 5/20 0.53
LMNA P02545 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136991 0.90 KMT2A (0.85) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL4466974 0.90 KMT2A (0.69) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL17179706 0.83 KMT2A (1.00) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL8126892 0.82 POLB (1.00) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL10924611 0.81 POLB (0.80) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL8128496 0.80 KDM4E (0.70) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL8146522 0.80 POLB (0.77) KMT2AMEN1ATMPOLBKDM4E
Hydrochloric Acid SCHEMBL9665606 0.80 POLB (0.77) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL8140905 0.79 POLB (0.76) KMT2AMEN1ATMPOLBKDM4E
SCHEMBL4475700 0.79 KDM4E (0.59) KMT2AMEN1ATMPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973773-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 2000-01-26 EP disclosed
WO-1998045293-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 1998-10-15 WO disclosed