SCHEMBL8147997

SCHEMBL8147997

COc1cc2c(cc1OC)-c1cc(Nc3ccccc3)nc(=O)n1CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 1.00
KMT2A Q03164 8/20 0.82
MEN1 O00255 4/20 0.81
POLB P06746 5/20 0.80
CASP6 P55212 1/20 0.80
CACNA1B Q00975 1/20 0.80
APBA1 Q02410 1/20 0.80
SIRT5 Q9NXA8 1/20 0.80
MAPT P10636 4/20 0.78
L3MBTL1 Q9Y468 2/20 0.78
ALDH1A1 P00352 8/20 0.74
HPGD P15428 6/20 0.74
HTT P42858 2/20 0.74
RXFP1 Q9HBX9 1/20 0.74
PDE4A P27815 1/20 0.73
GPR84 Q9NQS5 1/20 0.73
HSD17B10 Q99714 8/20 0.71
MAPK1 P28482 7/20 0.71
TSHR P16473 6/20 0.71
USP2 O75604 4/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8138318 0.89 KMT2A (0.80) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL8136991 0.88 KMT2A (0.85) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL8126892 0.86 POLB (1.00) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL8138535 0.86 KDM4E (0.76) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL10924611 0.85 POLB (0.80) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL9666833 0.85 POLB (0.80) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL8134020 0.84 GPR84 (1.00) KDM4EKMT2AMEN1POLBCASP6
Hydrochloric Acid SCHEMBL9665606 0.84 POLB (0.77) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL8146522 0.84 POLB (0.77) KDM4EKMT2AMEN1POLBCASP6
SCHEMBL8148567 0.84 POLB (0.82) KDM4EKMT2AMEN1POLBCASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973773-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 2000-01-26 EP claimed
WO-1998045293-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 1998-10-15 WO claimed
EP-0973773-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 2000-01-26 EP disclosed
WO-1998045293-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 1998-10-15 WO disclosed