SCHEMBL8148201

SCHEMBL8148201

O=C(Nc1ccccc1)Nc1ccc2[nH]nc(C3CCN4CCCCC4C3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 4/20 0.44
AURKA O14965 1/20 0.42
TTK P33981 1/20 0.42
PDPK1 O15530 2/20 0.41
BRD4 O60885 1/20 0.41
ITK Q08881 2/20 0.41
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41
FGFR1 P11362 1/20 0.41
FLT1 P17948 1/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
BTK Q06187 2/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
MAPK13 O15264 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8148939 0.97 ULK1 (0.44) ULK1AURKATTKPDPK1BRD4
SCHEMBL5906358 0.89 NPC1 (0.41) ULK1PDPK1ABL1BCRFGFR1
SCHEMBL5309301 0.87 JAK2 (0.53) ULK1AURKABRD4ITKJAK2
SCHEMBL5306459 0.85 HTR1D (0.42) AURKATTKBRD4
SCHEMBL8713578 0.83 SLC6A4 (0.52)
SCHEMBL5906388 0.83 JAK2 (0.36) ULK1TTKPDPK1ABL1BCR
SCHEMBL5302823 0.83 JAK2 (0.43) ULK1AURKAITKABL1BCR
SCHEMBL5312586 0.83 KDR (0.42) PDPK1ITKABL1BCRFGFR1
SCHEMBL5311332 0.82 JAK2 (0.56) ULK1ABL1BCRJAK2JAK1
SCHEMBL5311677 0.82 JAK2 (0.55) ULK1AURKABRD4ITKJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000006173-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed