SCHEMBL8148503

SCHEMBL8148503

Nc1c(O)c(Br)cc(F)c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.44
AKR1C2 P52895 3/20 0.40
AKR1C1 Q04828 3/20 0.40
AKR1C4 P17516 2/20 0.40
AKR1C3 P42330 2/20 0.40
PTPN1 P18031 3/20 0.37
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
PTPN2 P17706 1/20 0.34
PTPN6 P29350 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 2/20 0.33
CA12 O43570 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CA3 P07451 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21550525 0.83 HDAC1 (0.36) TTRHDAC1HDAC6CA1CA2
SCHEMBL8148621 0.82 TTR (0.48) TTRAKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL29133203 0.81 TTR (0.47) TTRAKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL24558455 0.80 KMT2A (0.35) TTRHDAC1HDAC6CA1CA2
SCHEMBL30929295 0.80 KMT2A (0.35) TTRHDAC1HDAC6CA1CA2
SCHEMBL23655038 0.77 TTR (0.47) TTRAKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL31426608 0.76 CA1 (0.37) HDAC1HDAC6CA1CA2CA9
SCHEMBL17541094 0.76 CA1 (0.41) TTRHDAC1HDAC6CA1CA2
SCHEMBL31728878 0.75 ALDH1A1 (0.37) AKR1C2AKR1C1CA1CA2TDP1
SCHEMBL20396360 0.75 TTR (0.48) TTRAKR1C2AKR1C1AKR1C4AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686145-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-01-26 EP disclosed
US-5883129-A Hydroxylated anthranilic acid derivatives ASTRA AKTIEBOLAG (SE) 1999-03-16 US disclosed
US-5523475-A New compounds AKTIEBOLAGET ASTRA (SE) 1996-06-04 US disclosed
CN-1121345-A New compounds ASTRA AB (SE) 1996-04-24 CN disclosed
EP-0686145-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1995-12-13 EP disclosed
WO-1994019316-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1994-09-01 WO disclosed