SCHEMBL8150342

SCHEMBL8150342

Cc1ccc(CN2C(=O)C(=O)N(CC(=O)O)C2=O)cc1

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.68
LMNA P02545 1/20 0.57
KMT2A Q03164 3/20 0.56
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MEN1 O00255 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
TP53 P04637 1/20 0.48
RAB9A P51151 1/20 0.48
LPAR1 Q92633 1/20 0.47
LPAR3 Q9UBY5 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8144324 0.85 KMT2A (0.58) MAPTKMT2AALDH1A1RAB9A
SCHEMBL8143584 0.85 KMT2A (0.76) MAPTKMT2AALDH1A1RAB9A
SCHEMBL8149613 0.84 MAPT (0.50) MAPTLMNAKMT2AHTTSMN1; SMN2
SCHEMBL8149456 0.84 KMT2A (0.56) MAPTLMNAKMT2AALDH1A1RAB9A
SCHEMBL8144325 0.84 KMT2A (0.56) MAPTKMT2AALDH1A1RAB9A
SCHEMBL9324908 0.82 KMT2A (0.72) MAPTKMT2AALDH1A1MEN1RAB9A
SCHEMBL8871897 0.81 KMT2A (0.56) MAPTKMT2AALDH1A1RAB9A
SCHEMBL8872045 0.80 ATM (0.55) MAPTKMT2AALDH1A1
SCHEMBL8873242 0.80 KMT2A (0.52) MAPTKMT2AALDH1A1HTTRAB9A
SCHEMBL8150317 0.80 KMT2A (0.52) MAPTKMT2AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6040326-A 3-deoxyglucosone production inhibitor NIPPON ZOKI PHARMACEUTICALS CO., LTD. (JP) 2000-03-21 US disclosed
EP-0855182-A1 3-Deoxyglucosone production inhibitor NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1998-07-29 EP disclosed
EP-0353198-B1 Parabanic acid derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO (JP) 1994-02-02 EP disclosed
US-4985453-A DIABETES TREATMENT NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1991-01-15 US disclosed
EP-0353198-A1 Parabanic acid derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1990-01-31 EP disclosed