SCHEMBL8871897

SCHEMBL8871897

O=C(O)CN1C(=O)C(=O)N(Cc2ccncc2)C1=O

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.56
MAPT P10636 2/20 0.49
RAB9A P51151 1/20 0.48
ALDH1A1 P00352 2/20 0.45
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
ELANE P08246 1/20 0.43
CTSG P08311 1/20 0.43
CMA1 P23946 1/20 0.43
CTRC Q99895 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8143584 0.85 KMT2A (0.76) KMT2AMAPTRAB9AALDH1A1F2
SCHEMBL8144324 0.82 KMT2A (0.58) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8872152 0.82 KMT2A (0.55) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8144325 0.81 KMT2A (0.56) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8149456 0.81 KMT2A (0.56) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8150342 0.81 MAPT (0.68) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8872045 0.80 ATM (0.55) KMT2AMAPTALDH1A1
SCHEMBL8872124 0.80 KMT2A (0.65) KMT2AMAPTALDH1A1
SCHEMBL8873242 0.77 KMT2A (0.52) KMT2AMAPTRAB9AALDH1A1
SCHEMBL8150317 0.77 KMT2A (0.52) KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681843-A ANTIDIABETIC; ALDOSE REDUCTASE INHIBITOR WITHOUT SUBSTANTIALLY INHIBITING ALDEHYDE REDUCATASE NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-10-28 US disclosed
EP-0718289-A1 Novel parabanic acid derivatives as aldose reductase inhibitors NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-06-26 EP disclosed