SCHEMBL8154087

SCHEMBL8154087

C=C(C)c1cccc(F)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
CES2 O00748 3/20 0.39
CES1 P23141 3/20 0.39
BCHE P06276 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
ALB P02768 1/20 0.36
ACHE P22303 1/20 0.36
GAA P10253 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
ALOX15 P16050 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HDAC4 P56524 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24832711 0.83 ESR1 (0.45) ESR1ESR2CES2CES1BCHE
SCHEMBL17040388 0.83 ESR1 (0.53) ESR1ESR2CES2CES1BCHE
SCHEMBL16959719 0.82 ESR1 (0.47) ESR1ESR2CES2CES1BCHE
SCHEMBL14040983 0.80 CES2 (0.56) CES2CES1BCHEALBGAA
SCHEMBL6862472 0.79 CES2 (0.52) CES2CES1BCHEACHEGAA
SCHEMBL30820836 0.79 CES2 (0.52) CES2CES1BCHEACHEGAA
SCHEMBL16956268 0.78 ESR1 (0.45) ESR1ESR2CES2CES1BCHE
SCHEMBL16957213 0.78 ESR1 (0.41) ESR1ESR2CES2CES1BCHE
SCHEMBL24832773 0.78 ESR1 (0.41) ESR1ESR2CES2CES1BCHE
SCHEMBL7135408 0.77 ESR1 (0.47) ESR1ESR2CES2CES1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4194452-A1 AROMATIC COMPOUND AND APPLICATION THEREOF IN ANTITUMOR DRUG Shanghai Zheye Biotechnology Co., Ltd. (CN) 2023-06-14 EP disclosed
WO-2023099648-A1 PYRAOLO- AND TRIAZOLO-AZINONE COMPOUNDS AND THEIR USES ASTRAZENECA AB (SE) 2023-06-08 WO disclosed
EP-4112606-A1 AROMATIC COMPOUND AND USE THEREOF IN PREPARING ANTINEOPLASTIC DRUGS Shanghai Zheye Biotechnology Co., Ltd. (CN) 2023-01-04 EP disclosed
EP-3835290-A1 OXADIAZOLINE COMPOUND OR SALT THEREOF, AGRICULTURAL OR HORTICULTURAL BACTERICIDE CONTAINING SAID COMPOUND, AND USE METHOD THEREFOR Nihon Nohyaku Co., Ltd. (JP) 2021-06-16 EP disclosed
WO-2008118849-A2 HIV-1 PROTEASE INHIBITORS UNIVERSITY OF MASSACHUSETTS (US) 2008-10-02 WO disclosed