SCHEMBL8154792

SCHEMBL8154792

COc1ccc2c(c1)C(CC(=O)O)=C(C)C2=Cc1ccc(Cl)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 6/20 0.64
PPARG P37231 14/20 0.62
CYP1A2 P05177 3/20 0.54
MAPT P10636 3/20 0.54
MAPK1 P28482 3/20 0.54
PTGS2 P35354 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
EGFR P00533 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
DRD1 P21728 1/20 0.54
PTGS1 P23219 1/20 0.54
OPRM1 P35372 1/20 0.54
PSEN1 P49768 1/20 0.54
PSEN2 P49810 1/20 0.54
APH1B Q8WW43 1/20 0.54
NCSTN Q92542 1/20 0.54
APH1A Q96BI3 1/20 0.54
PSENEN Q9NZ42 1/20 0.54
CYSLTR1 Q9Y271 1/20 0.54
PTGDR2 Q9Y5Y4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154789 1.00 RXRA (0.64) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL8154784 1.00 RXRA (0.64) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL30913437 0.97 RXRA (0.60) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL8681652 0.91 PPARG (0.64) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL8681649 0.91 PPARG (0.64) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL30913456 0.90 RXRA (0.58) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL8150041 0.89 PPARG (0.72) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL7147839 0.89 PPARG (0.72) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL8150043 0.89 PPARG (0.72) RXRAPPARGCYP1A2MAPTMAPK1
SCHEMBL12181845 0.89 RXRA (0.80) RXRAPPARGCYP1A2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028116-A Substituted condensation products of 1H-indenyl-hydroxyalkanes with aldehydes for neoplasia CELL PATHWAYS, INC. (US) 2000-02-22 US disclosed
US-5776962-A Lactone compounds for treating patient with precancerous lesions CELL PATHWAYS, INC. (US) 1998-07-07 US disclosed
US-5696159-A Lactone compounds for treating patients with precancerous lesions CELL PATHWAYS, INC. (US) 1997-12-09 US disclosed
US-4011332-A RODENTICIDE BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DT) 1977-03-08 US disclosed