Pyridine

Pyridine

SCHEMBL8158183

C=CCc1cc[nH]n1.c1ccncc1

nearest known ligand 0.31

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.31
NAPRT Q6XQN6 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479547 0.87
Pyridine SCHEMBL15010573 0.77 TSHR (0.35) TSHRNAPRTTDP1
Pyridine SCHEMBL27898466 0.76 PTPRA (0.33) TSHRNAPRTTDP1
Pyridine SCHEMBL27895501 0.73 CYP19A1 (0.36) TSHR
Pyridine SCHEMBL27297234 0.73 CYP1A2 (0.43) TDP1
Pyridine SCHEMBL28476914 0.71 L3MBTL1 (0.38) TDP1
Pyridine SCHEMBL28109232 0.70 TSHR (0.32) TSHRNAPRTTDP1
Pyridine SCHEMBL29208216 0.70 TDP1 (0.44) TDP1
Allylbenzene SCHEMBL28829822 0.70 MAOB (0.46) TSHRNAPRTTDP1
Pyridine SCHEMBL27261817 0.70 CYP3A4 (0.43) TSHRNAPRTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0594001-B1 Pyrazolo 4,3-c pyridines, a process for their preparation and their use as serotonin reuptake inhibitors AVENTIS PHARMA INC (US) 2000-08-16 EP disclosed
US-5428169-A Antidepressants, treating compulsive disorders, stuttering, trichotillomania HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-06-27 US disclosed
US-5380847-A Reaction of 1-methylpiperidine-4-hydrazine, ketone and titanium isopropoxide to form hydrazone HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1995-01-10 US disclosed
EP-0594001-A1 Pyrazolo 4,3-c pyridines, a process for their preparation and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-04-27 EP disclosed
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US disclosed
US-5264576-A Antiserotonin agents, antidepressants and obsessive-compulsive disorders HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-11-23 US disclosed